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Zosiyanasiyana Zilipo

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Zosakaniza Mbali

  • Itha kuthandiza antimalarial

Artemether CAS 71963-77-4 Artemisia Annua Extract

Artemether CAS 71963-77-4 Artemisia Annua Extract Image Featured

Tsatanetsatane wa Zamalonda

Zolemba Zamalonda

Zosakaniza Zosiyanasiyana N / A
Cas No 71963-77-4
Chemical Formula C16H26O5
Kulemera kwa maselo 298.37
EINECS no. 663-549-0
Malo osungunuka 86-88 ° C
Malo otentha 359.79 ° C (kuyerekeza molakwika)
Kuzungulira kwachindunji D19.5+171°(c=2.59inCHCl3)
Kuchulukana 1.0733 (kuyerekeza movutikira)
Index of refraction 1.6200 (chiyerekezo)
Zosungirako Kutentha kwapanyumba
Kusungunuka DMSO≥20mg/mL
Maonekedwe Ufa
Mawu ofanana ndi mawu Artemetherum/Artemtherin/Dihydroartemisininmethylether
Kusungunuka Zosungunuka mu Madzi
Magulu Zomera Zomera, Zowonjezera, Zaumoyo
Mapulogalamu Anti-malungo

Artemether ndi sesquiterpene lactone yomwe imapezeka mumizu yaArtemisia pachaka, omwe amadziwika kuti sweet chowawa.Ndi mankhwala amphamvu oletsa malungo omwe amagwiritsidwa ntchito pochiza ndi kupewa malungo.Artemisinin, kalambula bwalo wa artemether, idatulutsidwa koyamba kuchokera ku mbewuyi mu 1970s, ndipo kupezeka kwake kudapangitsa kuti wofufuza waku China, Tu Youyou, alandire Mphotho ya Nobel mu Medicine mu 2015.

Artemether amagwira ntchito powononga tizilombo toyambitsa malungo.Malungo amayamba ndi tizilombo toyambitsa matenda totchedwa Plasmodium, timene timapatsira anthu mwa kulumidwa ndi udzudzu waukazi wotchedwa Anopheles.Tizilombo toyambitsa matenda tikalowa m’thupi la munthu, timachulukirachulukira m’chiŵindi ndi m’maselo ofiira, ndipo zimenezi zimachititsa kutentha thupi, kuzizira, ndi zizindikiro zina zonga chimfine.Ngati sanalandire chithandizo, malungo akhoza kupha.

Artemether ndiwothandiza kwambiri polimbana ndi mitundu ina yosamva mankhwala ya Plasmodium falciparum, yomwe imachititsa kuti anthu ambiri azifa ndi malungo padziko lonse lapansi.Zimagwiranso ntchito polimbana ndi mitundu ina ya tizirombo ta Plasmodium toyambitsa malungo.Artemether nthawi zambiri amaperekedwa limodzi ndi mankhwala ena, monga lumefantrine, kuti achepetse chiopsezo cha kukana mankhwala.

Kupatula kugwiritsa ntchito ngati mankhwala oletsa malungo, artemether yapezekanso kuti ili ndi mankhwala ena.Kafukufuku wasonyeza kuti ali ndi anti-yotupa, anti-tumor, ndi anti-virus ntchito.Amagwiritsidwa ntchito pochiza nyamakazi, lupus, ndi matenda ena a autoimmune.Adafufuzidwanso kuti atha kuchiza COVID-19, ngakhale kafukufuku wochulukirapo akufunika kuti atsimikizire kugwira ntchito kwake.

Artemether nthawi zambiri imakhala yotetezeka komanso yololera bwino ikagwiritsidwa ntchito monga mwauzira.Komabe, monga mankhwala onse, angayambitse mavuto.Zotsatira zofala kwambiri za artemether ndi monga nseru, kusanza, chizungulire, ndi mutu.Nthawi zina, zimatha kuyambitsa zovuta zina, monga kugunda kwa mtima, khunyu, ndi kuwonongeka kwa chiwindi.

Pomaliza, artemether ndi mankhwala amphamvu oletsa malungo omwe asintha chithandizo cha malungo ndi kupewa.Kupezedwa kwake kwapulumutsa miyoyo yambiri ndipo kwachititsa kuti asayansi adziwike.Zina zake zochizira zimamupangitsa kukhala wodalirika wochizira matenda ena.Ngakhale zingayambitse mavuto, ubwino wake umaposa zoopsa zake zikagwiritsidwa ntchito moyang'aniridwa ndi achipatala.
Mafomu omwe amagwiritsidwa ntchito kwambiri ndi mapiritsi, makapisozi ndi jakisoni.Mitundu ya mankhwalawa ndi mankhwala oletsa malungo, ndipo chigawo chachikulu ndi artemether.The causative khalidwe la mapiritsi artemether anali woyera mapiritsi.Khalidwe la artemether capsule ndi capsule, zomwe zili mkati mwake ndi ufa woyera;Makhalidwe a mankhwala a jakisoni wa artemether ndi opanda utoto mpaka mafuta achikasu owala - ngati madzi.

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